A-366(5毫克)產品是A-366 is a potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC???= 3.3 nM). It displays >1000-fold selectivity for G9a/GLP over 21 other methyltransferases. A-366 has been shown to inhibit H3K9 methylation in prostate cancer PC3 cells with an IC???of 100 nM.