卵磷脂產品是Phloretin is a natural phenol which inhibits a variety of transporters. It inhibits the monocarboxylate transporters MCT1 and MCT2 (IC???= 28 and 14 μM, respectively), restricting the rapid transport of monocarboxylates like lactate and pyruvate across the plasma membrane. Phloretin also blocks the sodium/D-glucose cotransporter (Ki?= 86 μM) and the human concentrative nucleoside transporter 3 (Ki?= 32 μM). Blocks L-type Ca2??channels; activates Ca2?-activated K??channels in amphibian myelinated nerve fibers.
