BAZ2-ICR產品是BAZ2-ICR is a small molecule inhibitor of BAZ2A (Kd?= 109 nM; IC???= 130 nM) and BAZ2B (Kd?= 170 nM; IC50?= 180 nM) bromodomains. It displays 15-fold selectivity for binding BAZ2A/B over CECR2 and >100-fold selectivity over all other bromodomains.?BAZ2-ICR has been shown to displace BAZ2 bromodomains in living cells by demonstrating accelerated FRAP recovery at 1 μM in the BAZ2A FRAP assay.