D-螢光素,鈉鹽,StayBrite(500 ug)產(chǎn)品是Cell-permeable. A potent protein kinase C (PKC) inhibitor (IC?? = 7.9 nM). In vitro, discriminates between Ca2?-dependent and -independent isoforms of PKC; selectively inhibits PKCα and PKCβ1 (IC?? values are 2.3 and 6.2 nM respectively) but does not inhibit the activity of PKCδ, -ε, or -ζ (IC?? > 3uM).