PFI-1(1毫克)產(chǎn)品是PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4. In an AlphaScreen assay it has been shown to inhibit BRD2 bromodomain 2 and BRD4 bromodomain 1 with IC?? values of 98 nM and 0.22 uM, respectively.