ML243(5毫克)產(chǎn)品是ML-243 is a selective inhibitor of cancer stem cells. Displays 32-fold selective inhibition of a breast cancer stem cell-like cell line (EC?? = 2.0 uM) over a control (mammary epithelial) cell line (EC?? = 64 uM). It weakly antagonizes the adenosine A2A receptor (IC?? = 10 uM) and has no effect on 68 other targets commonly used in drug discovery for lead profiling.